Cinolazepam Information & Cinolazepam Links at HealthHaven.com

Not to be confused with clonazepam or camazepam.

Cinolazepam
Systematic (IUPAC) name


3-[9-chloro- 6-(2-fluorophenyl)- 4-hydroxy- 3-oxo- 2,5-diazabicyclo [5.4.0]undeca- 5,8,10,12- tetraen- 2-yl] propanenitrile
Identifiers
CAS number	75696-02-5
ATC code	N05CD13
PubChem	3033621
DrugBank	?
ChemSpider	2298251
Chemical data
Formula	C₁₈H₁₃Cl F N₃O₂
Mol. mass	357.8
SMILES	eMolecules & PubChem
Pharmacokinetic data
Bioavailability	90-100%
Metabolism	Hepatic
Half life	9 h^[1]
Excretion	Renal
Therapeutic considerations
Pregnancy cat.	?
Legal status	Unscheduled(US)
Routes	Oral
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Cinolazepam (marketed under the brand name Gerodorm)^[2] is a drug which is a benzodiazepine derivative. It possesses anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant properties. Due to its strong sedative properties, it is primarily used as an hypnotic.

Cinolazepam is not approved for sale in the United States or Canada.

[edit] See also

Benzodiazepine

[edit] References

^ Saletu, B.; G. Kindshofer, P. Anderer, J. Grunberger (1987). "Short-term sleep laboratory studies with cinolazepam in situational insomnia induced by traffic noise.". International Journal of Clinical Pharmacology Research 7 (5): 407–18. PMID 2889679.
^ Lannacher Romania (1999). "Gerodorm" (in Romanian). Produse Gerot inregistrate in Romania. http://www.lannacher.ro/gerodorm.html. Retrieved 17 August 2006.

[edit] External links

Inchem.org - Cinolazepam

v • d • e Benzodiazepines (N05BA, N05CD)

1,4-Benzodiazepines	Bromazepam • Camazepam • Chlordiazepoxide • Cinolazepam • Clonazepam • Clorazepate • Cyprazepam • Delorazepam • Diazepam • Doxefazepam • Elfazepam • Ethyl carfluzepate • Ethyl dirazepate • Ethyl loflazepate • Fletazepam • Fludiazepam • Flunitrazepam • Flurazepam • Flutemazepam • Flutoprazepam • Fosazepam • Gidazepam • Halazepam • Iclazepam • Lopirazepam • Lorazepam • Lormetazepam • Meclonazepam • Medazepam • Menitrazepam • Metaclazepam • Nimetazepam • Nitrazepam • Nitrazepate • Nordazepam • Oxazepam • Phenazepam • Pinazepam • Pivoxazepam • Prazepam • Proflazepam • Quazepam • QH-II-66 • Reclazepam • Sulazepam • Temazepam • Tetrazepam • Uldazepam

1,5-Benzodiazepines	Arfendazam • Clobazam • Lofendazam • Triflubazam

2,3-Benzodiazepines	Girisopam • GYKI-52466 • GYKI-52895 • Nerisopam • Tofisopam

Triazolobenzodiazepines	Adinazolam • Alprazolam • Estazolam • Triazolam

Imidazobenzodiazepines	Bretazenil • Climazolam • Flumazenil • Imidazenil • L-655,708 • Loprazolam • Midazolam • PWZ-029 • Ro15-4513 • Ro48-6791 • Sarmazenil • SH-053-R-CH3-2′F

Oxazolobenzodiazepines	Cloxazolam • Flutazolam • Haloxazolam • Mexazolam • Oxazolam

Thienodiazepines	Brotizolam • Ciclotizolam • Clotiazepam • Etizolam

Pyridodiazepines	Zapizolam • Lopirazepam

Pyrazolodiazepines	Ripazepam • Zolazepam • Zomebazam

Pyrrolodiazepines	Premazepam

Benzodiazepine Prodrugs	Avizafone • Rilmazafone

Others	Bentazepam • Devazepide • Ketazolam • Razobazam • Tifluadom

Hypnotics/Sedatives (N05C)

GABA_A receptor

Barbiturates

Ultrashort-acting	Methohexital • Thiamylal • Thiopental

Short/intermediate- acting	Allobarbital • Amobarbital • Aprobarbital • Butobarbital • Pentobarbital • Secobarbital • Talbutal

Long-acting	Barbital • Mephobarbital • Phenobarbital

Ungrouped	Cyclobarbital • Ethallobarbital • Heptabarbital • Hexobarbital • Proxibarbal • Reposal • Vinylbital • Vinbarbital

Benzodiazepines

Short-acting	Brotizolam • Cinolazepam • Doxefazepam • Loprazolam • Midazolam • Triazolam

Intermediate-acting	Estazolam • Flunitrazepam • Lormetazepam • Nimetazepam • Temazepam

Long-acting	Flurazepam • Flutoprazepam • Nitrazepam • Quazepam

Dialkylphenols

Fospropofol • Propofol • Thymol

Nonbenzo-
diazepines

CL-218,872 • Eszopiclone • Indiplon • Necopidem • Pazinaclone • ROD-188 • Saripidem • Suproclone • Suriclone • SX-3228 • U-89843A • U-90042 • Zaleplon • Zolpidem • Zopiclone

Piperidinediones

Glutethimide • Methyprylon • Pyrithyldione • Piperidione

Quinazolinones

Afloqualone • Cloroqualone • Diproqualone • Etaqualone • Mebroqualone • Mecloqualone • Methaqualone • Methylmethaqualone

Neuroactive
steroids

Acebrochol • Allopregnanolone • Alphadolone • Alphaxolone • Ganaxolone • Hydroxydione • Minaxolone • Org 20599 • Tetrahydrodeoxycorticosterone

Alpha-2 adrenergic
receptor

Alpha-adrenergic agonists

4-NEMD • Clonidine • Dexmedetomidine • Lofexidine • Medetomidine • Romifidine • Tizanidine • Xylazine

Melatonin receptor

Melatonin

Agomelatine • Melatonin • Ramelteon • Tasimelteon • Circadin

Histamine receptor &
Acetylcholine receptor

Antihistamines &
Anticholinergics

Amitriptyline • Dimenhydrinate • Doxylamine • Hydroxyzine • Diphenhydramine • Bromodiphenhydramine • Carbinoxamine • Doxepin • Orphenadrine • Mianserin • Mirtazapine • Nefazodone • Niaprazine • Phenyltoloxamine • Propiomazine • Pyrilamine • Scopolamine • Trazodone

GABA_B receptor /
GHB receptor

GHB Type

1,4-Butanediol • Aceburic acid • GABOB • GHB (Sodium Oxybate, Xyrem®) • GBL • gamma-Valerolactone

Orexin receptors

Orexin antagonists

Almorexant • SB-334,867 • SB-408,124 • SB-649,868 • TCS-OX2-29

Other receptors/
ungrouped

Aldehydes	Acetylglycinamide chloral hydrate • Chloral hydrate • Chloralodol • Dichloralphenazone • Paraldehyde • Petrichloral

Alkynes	Centalun • Ethchlorvynol • Ethinamate • Hexapropymate • Methylpentynol

Carbamates	Meprobamate • Carisoprodol • Tybamate • Methocarbamol • Procymate

Other	2-Methyl-2-butanol • Acecarbromal • Acetophenone • Apronal • Bromides • Bromisoval • Carbromal • Chloralose • Clomethiazole • Embutramide • Etomidate • Evoxine • Fenadiazole • Gaboxadol • Loreclezole • Mephenoxalone • Sulfonmethane • Trichloroethanol • Triclofos • Valerian • Valnoctamide

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Retrieved from "http://en.wikipedia.org/wiki/Cinolazepam"

Categories: Benzodiazepines | Hypnotics | Sedative stubs